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原料药及其中间体

序号 产品名称 英文名称 CAS No.
1 阿法替尼 Afatinib 850140-72-6
2 反式-4-二甲基胺基巴豆酸盐酸盐 trans-4-Dimethylaminocrotonic acid hydrochloride 848133-35-7
3 (S)-(+)-3-羟基四氢呋喃 (S)-(+)-3-Hydroxytetrahydrofuran 86087-23-2
4 (R)-(-)-3-羟基四氢呋喃 (R)-(-)-3-Hydroxytetrahydrofuran 86087-24-3
5 7-氯-6-硝基喹唑啉-4-酮 6-Nitro-7-Chloro-4-HydroxyQuinazoline 53449-14-2
6 7-氟-6-硝基-4-羟基喹唑啉 7-Fluoro-6-nitro-4-hydroxyquinazoline 162012-69-3
7 4-[(3-氯-4氟)氨基]-6-硝基-7-氟-喹唑啉氨 4-Quinazolinamine, N-(3-chloro-4-fluorophenyl)-7-fluoro-6-nitro- 162012-67-1
8 阿哌沙班 Apixaban 503612-47-3
9 [(4-甲氧基苯基)肼基]氯乙酸乙酯 Acetic acid, 2-chloro-2-[2-(4-methoxyphenyl)hydrazinylidene], ethyl ester 27143-07-3
10 5,6-二氢-3-(4-吗啉基)-1-(4-硝基苯基)-2(1H)-吡啶酮 3-(4-Morpholinyl)-1-(4-nitrophenyl)-5,6-dihydro-2(1H)-pyridinone 503615-03-0
11 4,5,6,7-四氢-1-(4-甲氧基苯基)-6-(4-硝基苯基)-7-氧代-1H-吡唑并[3,4-C]吡啶-3-羧酸乙酯 4,5,6,7-Tetrahydro-1-(4-methoxyphenyl)-6-(4-nitrophenyl)-7-oxo-1H-pyrazolo[3,4-c]pyridine-3- 536759-91-8
12 1-(4-甲氧基苯基)-7-氧代-6-[4-(2-氧代哌啶-1-基)苯基]-4,5,6,7-四氢-1H-吡唑并[3,4-C]吡啶-3-羧酸乙酯 ethyl 1-(4-methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H- 503614-91-3
13 5,6-二氢-3-(4-吗啉基)-1-[4-(2-氧代-1-哌啶基)苯基]-2(1H)-吡啶酮 5,6-Dihydro-3-(4-morpholinyl)-1-[4-(2-oxo-1-piperidinyl)phenyl]-2(1H)-pyridinone 545445-44-1
14 贝达喹啉 Bedaquiline 843663-66-1
15 3-(二甲基氨基)-1-(萘-1-基)-1-丙酮盐酸盐 3-dimethylamino-1-(naphthalen-1-yl)propan-1-one hydrochloride 5409-58-5
16 3-苄基-6-溴-2-甲氧基喹啉 3-benzyl-6-bromo-2-methoxyquinoline 654655-69-3
17 盐酸苯达莫斯汀 Bendamustine hydrochloride 3543-75-7
18 4-(1-甲基-5-氨基-1H-苯并咪唑-2-基)丁酸乙酯 4-(5-amino-1-methyl-1H-benzoimidazol-2-yl)-butyric acid ethyl ester 3543-73-5
19 瑞替加滨 Retigabine 150812-12-7
20 瑞替加滨二盐酸盐 Ethyl [2-amino-4-[[(4-fluorophenyl)methyl]amino]phenyl]carbamatedihydrochloride 150812-13-8
21 2-氨基-5-(4-氟苄氨基)硝基苯 2-Amino-5-[(4-fluorobenzyl)amino]-1-nitrobenzene 150812-21-8
22 索拉菲尼 Sorafenib tosylate 284461-73-0
23 N-甲基-4-氯-2-吡啶甲酰胺 N-Methyl-4-chloropyridine-2-carboxamide 220000-87-3
24 1-氯-3,5-二-O-对甲苯甲酰基-2-脱氧-D-呋喃核糖 1-Chloro-3,5-di-O-toluoyl-2-deoxy-D-ribofuranose 3601-89-6
25 4-氨基-3-氟苯酚 4-Amino-3-fluorophenol 399-95-1
26 4-氯-3-三氟甲基异氰酸苯酯 4-Chloro-3-(trifluoromethyl)phenyl isocyanate 327-78-6
27 对氨基酚 4-Aminophenol 123-30-8
28 沙格列汀 Saxagliptin 361442-04-8
29 (1S,3S,5S)-3-(氨基羰基)-2-氮杂双环[3.1.0]己烷-2-甲酸叔丁酯 (1S,3S,5S)-3-(Aminocarbonyl)-2-azabicyclo[3.1.0]hexane-2-carboxylic acid tert-butyl ester 361440-67-7
30 N-叔丁氧羰基-3-羟基-1-金刚烷基-D-甘氨酸 (alphaS)-alpha-[[(1,1-Dimethylethoxy)carbonyl]amino]-3-hydroxytricyclo[3.3.1.13,7]decane-1- 361442-00-4
31 维达列汀 Vildagliptin 274901-16-5
32 L-脯氨酰胺 Prolinamide 7531-52-4
33 3-胺基-1-金刚烷醇 1-Amino-3-adamantanol 702-82-9
34 (2S)-N-氯乙酰基-2-氰基四氢吡咯 (S)-2-cyanopyrrolidine-1-carbonyl chloride 207557-35-5
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